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1. H1 antagonist - Wikipedia
Link: https://en.wikipedia.org/wiki/H1_antagonist
Description:
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2. Histamine H1 Antagonists | DrugBank Online
Link: https://go.drugbank.com/categories/DBCAT000665
Description: Dr. Himanshu J. Vats
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3. H1 antagonist - Wikipedia
Link: https://en.wikipedia.org/wiki/H1_antagonist
Description: H1-antihistamines are clinically used in the treatment of histamine-mediated allergic conditions. These indications may include: Allergic rhinitisAllergic conjunctivitisAllergic dermatological conditions (contact dermatitis)Rhinorrhea (runny nose)UrticariaAngioedemaDiarrheaPruritus (atopic dermatitis, … See more
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4. Histamine H1 Antagonists | DrugBank Online
Link: https://go.drugbank.com/categories/DBCAT000665
Description: WEB1031 rows · Description. Drugs that selectively bind to but do not activate histamine H1 …
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5. Explore further
Link: https://go.drugbank.com/drugs/DB00283
Description:
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6. Antihistamines - StatPearls - NCBI Bookshelf
Link: https://www.ncbi.nlm.nih.gov/books/NBK538188/
Description: WEBJul 10, 2023 · First-generation antihistamines easily cross the blood-brain barrier into the central nervous system and antagonize H-1 receptors, …
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7. Antiemetic Histamine H1 Receptor Blockers - StatPearls
Link: https://www.ncbi.nlm.nih.gov/books/NBK533003/
Description: WEBMar 7, 2023 · Summarize the mechanism of action of H1 receptor blockers. Identify the approved indications for H1 receptor blockers. Review the … Author: Travis S. Schaefer, Patrick M. Zito Publish Year: 2019
Author: Travis S. Schaefer, Patrick M. ZitoPublish Year: 2019
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8. Histamine receptors, agonists, and antagonists in health …
Link: https://pubmed.ncbi.nlm.nih.gov/34225942/
Description: WEBH1 receptor antagonists have been used to treat insomnia, but its use requires precautions due to potential side effects. H2 receptor antagonists have shown efficacy … Author: Pertti Panula Publish Year: 2021
Author: Pertti PanulaPublish Year: 2021
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9. Diphenhydramine - StatPearls - NCBI Bookshelf
Link: https://www.ncbi.nlm.nih.gov/books/NBK526010/
Description: WEBJul 10, 2023 · Diphenhydramine mainly works through antagonizing the H1 (histamine 1) receptor, although it has other mechanisms of action as well. [1] The H1 receptor is located on respiratory smooth muscles, vascular …
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10. Advances in H 1 -Antihistamines - The New England …
Link: https://www.nejm.org/doi/full/10.1056/NEJMra033121
Description: WEBNov 18, 2004 · Through the H 1 -receptor, histamine has proinflammatory activity and is involved in the development of several aspects of antigen-specific immune response, including the maturation of...
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11. Molecular mechanism of antihistamines recognition and …
Link: https://www.nature.com/articles/s41467-023-44477-4
Description: WEBJan 2, 2024 · Antihistamines that target the histamine H 1 receptor (H 1 R) have been widely used to relieve the symptoms of allergy and inflammation.
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12. The Pharmacology and Use of H 1 -Receptor-Antagonist …
Link: https://www.nejm.org/doi/full/10.1056/NEJM199406093302307
Description: WEBJun 9, 1994 · Histamine H 1 antagonists are highly selective for H 1 receptors, having little effect on H 2 or H 3 receptors. First-generation H 1 -receptor antagonists may also activate muscarinic...
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13. Real-world evidence for improved outcomes with …
Link: https://www.nature.com/articles/s41392-021-00689-y
Description: WEBJul 14, 2021 · (ii) Histamine H 2 receptor antagonists (H2RA) competitively bind the H2R, a type of G-protein coupled receptor (GPCR), 1 and block the natural stimulation of its …